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カタログ番号	製品名	別名	ターゲット
T36816	S-trityl-L-Cysteine	STLC	Kinesin
	S-trityl-L-Cysteine is a non-natural amino acid and an inhibitor of Eg5, also known as KSP and Kif11, a mitotic kinesin necessary for mitotic spindle formation. S-trityl-L-Cysteine inhibits the ATPase activity of Eg5 in ...		Kinesin
T9636	Dalpiciclib	SHR-6390	CDK
	Dalpiciclib (SHR-6390) is a highly selective, orally bioavailable, and comparable potency inhibitor of CDK4 and CKD6 with IC50s of 12.4 nM and 9.9 nM, respectively. Dalpiciclib exerts potent antitumor activity in esophag...		CDK
T0431	Abexinostat	CRA 24781,PCI24781,PCI-24781,PCI 24781,CRA 024781	HDAC
	PCI-24781 (Abexinostat (PCI24781)) is a new pan-HDAC inhibitor mainly targeting HDAC1 (Ki: 7 nM), also have moderate inhibitory for HDACs 2, 3, 6, and 10 and greater than 40-fold selectivity against HDAC8. Phase 1/2.		HDAC
T10342	Antitumor agent-2		Others
	Antitumor agent-2 has anti-inflammatory and anti-tumor activity and can be used to study cancer.		Others
T12692	RAS GTPase inhibitor 1		Raf
	RAS GTPase inhibitor 1 is a RAS GTPase inhibitor with potential antitumor activity.		Raf
T7611	ODM-203		VEGFR , FGFR
	ODM-203, a Selective Inhibitor of FGFR and VEGFR, Shows Strong Antitumor Activity, and Induces Antitumor Immunity		VEGFR , FGFR
T72027	6-Methyl-3-pyridinecarboxaldehyde	6-Methoxynicotinaldehyde
	6-Methyl-3-pyridinecarboxaldehyde (6-Methoxynicotinaldehyde) has partial antitumor activity.
T13799	NQO1 substrate		NADPH
	NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research.		NADPH
T6821	Dp44mT		Apoptosis , Others , Ferroptosis
	Dp44mT, a effective iron chelator, has selective antitumor activity.		Apoptosis , Others , Ferroptosis
T35262	YM 534	YM-534,YM534	Others
	YM 534 has antitumor activity and platelet aggregation activity, inhibits photoaffinity labeling of deglycosylated P-glycoprotein, and can be used to study leukemia.		Others
T9998	MIND4-19		Sirtuin
	MIND4-19 is an inhibitor of SIRT2 with antitumor activity.		Sirtuin
T16913	Sotirimod	R850,S-30594	Virus Protease
	Sotirimod（R850） is a novel immunomodulator with antitumor and antiviral activity for the study of actinic keratoses.		Virus Protease
T28189	Nortopixantrone HCl	BBR3438,Nortopixantrone hydrochloride,BBR-3438	Others
	Nortopixantrone HCl (BBR 3438) is a novel 9-azacyclonopyrazole that shows antitumor activity in a human prostate cancer model.		Others
T16551	Pladienolide B		Apoptosis
	Pladienolide B is a potent spliceosome inhibitor, a macrolide isolated from Streptomyces obtusususus Mer-12, which targets the SF3B1 subunit of the spliceosome.Pladienolide B exerts its antitumor effects by inhibiting pr...		Apoptosis
T27583	IDD388	IDD-388,IDD 388	DNA/RNA Synthesis
	IDD388 is a selective and potent aldose reductase (ALR2) inhibitor with antitumor activity that inhibits the ALR1 receptor.		DNA/RNA Synthesis
T10276L	AKT Kinase Inhibitor HCl	AKT Kinase Inhibitor HCl(842148-40-7 Free base)	Akt
	AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity.		Akt
T15653	Ketocaine	Rec 7-0518	Others
	Ketocaine（Rec 7-0518） is a local anesthetic commonly used in animal experiments with potential antitumor activity for pain relief.		Others
TNU0123	5-Methoxyuridine	Mo5U	Apoptosis
	5-Methoxyuridine (Mo5U) is a purine nucleoside analog with a broad spectrum of antitumor activity, targeting malignant tumors of the inert lymphatic system and inducing apoptosis.5-Methoxyuridine's anticancer mechanism i...		Apoptosis
T16716	Rabacfosadine	VDC-1101,GS-9219	Others
	Rabacfosadine (GS-9219) is a novel prodrug of PMEG, an acyclic nucleotide phosphonate, with antitumor activity for the study of lymphoma.		Others
T17032	Telratolimod	MEDI9197,3M-052	TLR
	Telratolimod (MEDI9197) is a toll-like receptors 7/8 agonist. It has an antitumor activity.		TLR
T23647	Zindoxifene	D 16726	Estrogen/progestogen Receptor
	Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer.		Estrogen/progestogen Receptor
T9629	BRD4 Inhibitor-24		Epigenetic Reader Domain
	BRD4 Inhibitor-24 is a BRD4 small molecule inhibitor with antitumor activity.		Epigenetic Reader Domain
T7969	Dipyrithione		Others
	Dipyrithione appears to have novel cytotoxicity and potent broad-spectrum antitumor activity		Others
T14894	CC-90003		ERK
	CC-90003 is a selective inhibitor of ERK 1/2. It has antitumor activity.		ERK
T8523	ILK-IN-3		Integrin
	ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.		Integrin
T67735	Auristatin23		Others
	Auristatin23 is an Antitumor agent. Auristatin23 exhibits antiproliferative activity on tumor cell lines.		Others
T14380	AZD7507		CSF-1R , HER , Sodium Channel
	AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.		CSF-1R , HER , Sodium Channel
T24818	Sparfosic Acid	NSC224131,NSC-224131,Acide sparfosique,N-Phosphonacetyl-L-aspartate,NSC 224131	Apoptosis
	Sparfosic Acid (Acide sparfosique) is an aspartate carbamoyltransferase inhibitor with antitumor activity and can be used to study advanced renal cell carcinoma.		Apoptosis
T16788	Rosabulin	STA 5312	Others , Microtubule Associated
	v Rosabulin (STA 5312) is an orally active microtubule inhibitor with potency. Rosabulin inhibits microtubule assembly and has broad-spectrum antitumor activity.		Others , Microtubule Associated
T78631	Ac-YVAD-AOM		Caspase
	Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.		Caspase
T1910	Ansamitocin P 3'	Maytansinol butyrate,Ansamitocin P-3,Antibiotic C 15003P3'	Microtubule Associated
	Ansamitocin P 3' (Maytansinol butyrate) is an antibody-drug conjugate cytotoxin with antitumor activity.		Microtubule Associated
T1775	GSK503		Histone Methyltransferase
	GSK-503, a potent EZH2 inhibitor, has potential antitumor activity.		Histone Methyltransferase
T12894	SGN-2FF		Others
	SGN-2FF is an oral fucosylation inhibitor and inhibits fucosyltransferase activity, and has antitumor activity.		Others
T23911	CPS-11	CPS11,CPS 11,N-(Hydroxymethyl)thalidomide	Dehydrogenase , NF-κB , Reactive Oxygen Species
	CPS-11 (N-(Hydroxymethyl)thalidomide) is a Thalidomide analogue that has significant antitumor activity and exhibits a wider range of activity and highly potent effects on the MM (multiple myeloma) cell line.		Dehydrogenase , NF-κB , Reactive Oxygen Species
T26625	AN-019	NRC-AN-019,NRC-019	Bcr-Abl
	AN-019 (NRC-019) is a Bcr-Abl kinase inhibitor with antitumor activity for the study of chronic myelogenous leukemia (CML) and breast cancer.		Bcr-Abl
T8216	T-1101 tosylate	TAI-95 tosylate	Apoptosis , Microtubule Associated
	T-1101 tosylate (TAI-95 tosylate) is an inhibitor of Hec1/Nek2, with antitumor activity.		Apoptosis , Microtubule Associated
T10678	Carboxypeptidase G2 (CPG2) Inhibitor	CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor	Carboxypeptidase
	Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.		Carboxypeptidase
T67785	ABI-1968		Antiviral
	ABI-1968 has antiviral and antitumor activity and can be used to study immune system diseases.		Antiviral
T30745L	Carboxy-pyridostatin 2HCl	Carboxy-pyridostatin 2HCl(1417638-60-8 Free base）	DNA
	Carboxy-pyridostatin 2HCl has potential antitumor activity with high affinity for DNA at DNA G4s.		DNA
T77512	1H-Benzimidazole-6-carboxamide, N-[3-(aminocarbonyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-		Others
	1H-Benzimidazole-6-carboxamide, N-[3-(aminocarbonyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]- may have antitumor activity.		Others
T11190	EMT inhibitor-1		Wnt/beta-catenin
	EMT inhibitor-1 is an inhibitor of Hippo, Wnt signaling and TGF- macrophages (TGF-) with antitumor activity.		Wnt/beta-catenin
T6810	CPI-360	Synonym 2,CPI 360,CPI360	Apoptosis , Histone Methyltransferase
	CPI-360 is a small molecule EZH2 inhibitor (IC50: 0.002 μM, EC50: 0.080 μM) that shows antitumor activity in an EZH200-dependent tumor xenograft model.		Apoptosis , Histone Methyltransferase
T6210	Pifithrin-μ	PFTμ,NSC 303580,2-Phenylethynesulfonamide	HSP , p53 , Autophagy
	Pifithrin-μ (NSC-303580) is an inhibitor of p53 and HSP70, with neuroprotective and antitumor activity.		HSP , p53 , Autophagy
T27138	Declopramide	OXI-104,IMO-B,3-Chloroprocainamide	Apoptosis
	Declopramide (OXI-104) is a novel chemosensitizer with antitumor activity that induces apoptosis and can be used to study colorectal cancer and inflammatory bowel disease.		Apoptosis
T11872L	LMP744 hydrochloride	NSC706744 hydrochloride,MJ-III65 hydrochloride	Topoisomerase
			Topoisomerase
T9593	Senaparib	IMP4297	PARP
	Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.		PARP
T15597L	ISA-2011B-P2
	ISA-2011B-P2 is a stereoisomer of ISA-2011B, a potent PIP5K1α inhibitor with antitumor activity.
T27257	EMD-503982	EMD503982,EMD 503982	Factor Xa
	EMD-503982 is a potential Factor Xa and Factor VIIa inhibitor with potential anticancer and antitumor activity for the study of thromboembolic and neurological disorders.		Factor Xa
T67945	WAY-620473		PARP
	WAY-620473 is a potent PARP-1 inhibitor with antitumor activity and alters eukaryotic lifespan.		PARP
T7819	TAS0728		EGFR , HER
	TAS0728 is a HER2 inhibitor, with antitumor activity		EGFR , HER

Compounds

Synonym: CRA 24781,PCI24781,PCI-24781,PCI 24781,CRA 024781

RAS GTPase inhibitor 1

6-Methyl-3-pyridinecarboxaldehyde

T72027

Synonym: 6-Methoxynicotinaldehyde

Target: Apoptosis, Others, Ferroptosis

YM 534

T35262

Synonym: YM-534,YM534

Synonym: R850,S-30594

Target: Virus Protease

Nortopixantrone HCl

T28189

Synonym: BBR3438,Nortopixantrone hydrochloride,BBR-3438

Synonym: IDD-388,IDD 388

Target: DNA/RNA Synthesis

AKT Kinase Inhibitor HCl

T10276L

Synonym: AKT Kinase Inhibitor HCl(842148-40-7 Free base)

Synonym: VDC-1101,GS-9219

Target: Others

Telratolimod

T17032

Synonym: MEDI9197,3M-052

Target: Estrogen/progestogen Receptor

BRD4 Inhibitor-24

T9629

Synonym:

Target: Epigenetic Reader Domain

Target: CSF-1R, HER, Sodium Channel

Sparfosic Acid

T24818

Synonym: NSC224131,NSC-224131,Acide sparfosique,N-Phosphonacetyl-L-aspartate,NSC 224131

Target: Others, Microtubule Associated

Synonym: Maytansinol butyrate,Ansamitocin P-3,Antibiotic C 15003P3'

Target: Microtubule Associated

GSK503

T1775

Synonym:

Target: Histone Methyltransferase

Synonym: CPS11,CPS 11,N-(Hydroxymethyl)thalidomide

Target: Dehydrogenase, NF-κB, Reactive Oxygen Species

AN-019

T26625

Synonym: NRC-AN-019,NRC-019

Target: Bcr-Abl

T-1101 tosylate

T8216

Synonym: TAI-95 tosylate

Target: Apoptosis, Microtubule Associated

Carboxypeptidase G2 (CPG2) Inhibitor

T10678

Synonym: CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor

Target: Carboxypeptidase

Carboxy-pyridostatin 2HCl

T30745L

Synonym: Carboxy-pyridostatin 2HCl(1417638-60-8 Free base）

Target: DNA

1H-Benzimidazole-6-carboxamide, N-[3-(aminocarbonyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-

Target: Wnt/beta-catenin

CPI-360

T6810

Synonym: Synonym 2,CPI 360,CPI360

Target: Apoptosis, Histone Methyltransferase

Pifithrin-μ

T6210

Synonym: PFTμ,NSC 303580,2-Phenylethynesulfonamide

Target: HSP, p53, Autophagy

Declopramide

T27138

Synonym: OXI-104,IMO-B,3-Chloroprocainamide

Target: Apoptosis

LMP744 hydrochloride

T11872L

Synonym: NSC706744 hydrochloride,MJ-III65 hydrochloride

Target: Topoisomerase

Synonym: EMD503982,EMD 503982

カタログ番号	製品名	別名	ターゲット
T6S0923	Hypericin	Hypericine,Cyclosan	Apoptosis , Antiviral , Influenza Virus , Tyrosine Kinases , Antibacterial , PKC
	1. Hypericin (Cyclosan) has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoamine oxidase enzyme. 4. Hypericin inhibits RANKL...
T67047	2-Acetyl-3-ethylpyrazine		Endogenous Metabolite
	2-Acetyl-3-ethylpyrazine has antitumor activity.		Endogenous Metabolite
T3S1457	Palmaturbine	Palmatrubin,Palmatrubine	Others
	Palmaturbine (Palmatrubine) shows high antitumor activity.		Others
TN7217	4,6-Benzilidine-D-Glucose
	4,6-Benzilidine-D-Glucose is a clinical antitumor compound showing antitumor activity in rats with chemically induced hepatocellular carcinoma.
T11354	Gambogellic acid
	Gambogellic acid is an xanthone compound obtained from Garcinia cambogia and processed Gambog, is antitumor activity and cytotoxicity.
T2736	Sodium Demethylcantharidate	Sodium norcantharidin	Others , Endogenous Metabolite
	Sodium Demethylcantharidate (Sodium norcantharidin) is extracted from Mylabris phqlarata pallas and has potent antitumor activity.		Others , Endogenous Metabolite
TN7250	Torachrysone Triglucoside	1-[8-[(O-β-D-Glucopyranosyl-(1→3)-O-β-D-glucopyranosyl-(1→6)-β-D-glucopyranosyl)oxy]-1-hydroxy-6-methoxy-3-methyl-2-naphthalenyl]ethanone	Others
	Torachrysone Triglucoside is a glucoside isolated from cassia seeds with potential antitumor activity.		Others
T1687	Doxycycline	Vibramycin,Doxiciclina,Doxytetracycline,Doxycyclinum	MMP , ribosome , Antibacterial , Antibiotic , Parasite
	Doxycycline (Doxiciclina) belongs to the tetracycline class of antibiotics and is a broad-spectrum metalloproteinase (MMP) inhibitor with oral activity. Doxycycline has antibacterial activity and antitumor activity.		MMP , ribosome , Antibacterial , Antibiotic , Parasite
T5581	6-(γ,γ-Dimethylallylamino)purine	N6-(2-lsopentenyl)adenine,Triacanthine	Others
	6-(γ,γ-Dimethylallylamino)purine (Triacanthine), which is a plant growth substance, shows hypertensive and antitumor activity, also cardiotonic, antispasmodic and a respiratory analeptic.		Others
T3878	Raddeanin A	NSC382873,Anemodeanin A,Raddeanin R3	Apoptosis , HDAC
	Raddeanin A (NSC-382873) has moderate inhibitory activity against histone deacetylases (HDACs). Raddeanin A has high antiangiogenic potency, antitumor activity.		Apoptosis , HDAC
T2217	Cephalomannine	Baccatin III	Microtubule Associated
	Cephalomannine (Baccatin III) is a taxol derivative obtained from Taxus yunnanensis with antitumor activity.		Microtubule Associated
T1687L	Doxycycline (hyclate)	Doxycycline hydrochloride hemiethanolate hemihydrate,WC2031,Doxycycline hyclate	MMP , ribosome , Antibacterial , Antibiotic
	Doxycycline hyclate (WC2031) belongs to the tetracycline class of antibiotics and is a broad-spectrum metalloproteinase (MMP) inhibitor with oral activity. Doxycycline hyclate has antibacterial activity and antitumor act...		MMP , ribosome , Antibacterial , Antibiotic
T5S0662	Gelsemine	Gelsemin	Antioxidant
	1. Gelsemine (Gelsemin) has antitumor activity. 2. Gelsemine has anti-oxidative activity. 3. Gelsemine has anti-hyperlipidemic activity. 4. Gelsemine has marked antinociception in inflammatory, neuropathic and bone cance...		Antioxidant
T6S1844	Tenacissoside H	Tenacissimoside C	Others
	Tenacissoside H (Tenacissimoside C) has antitumor activity on esophageal cancer through arresting cell cycle and regulating PI3K/Akt-NF-κB transduction cascade.		Others
T3819	Ursolic acid acetate	Acetylursolic acid,3-Acetylursolic Acid	AChE
	Ursolic acid acetate (Acetylursolic acid) has cytotoxic activity, antimalarial activity, antitumor and anticancer activities. Acetylursolic acid has NO production inhibitory activities. Acetylursolic acid has inhibition ...		AChE
T1508	Decitabine	Dacogen,NSC 127716,Deoxycytidine,5-Aza-2'-deoxycytidine	Apoptosis , Nucleoside Antimetabolite/Analog , DNA Methyltransferase
	Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity. Decitabine has antitumor activity and antimetabolic activity. Decitabine induces cell cycle arrest and apoptosis...
TC0025	Testosterone acetate	NSC523836,NSC-523836,NSC 523836	Others
	Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.		Others
TN1008	Psoralenoside		CaMK , Calcium Channel , Histamine Receptor
	Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.		CaMK , Calcium Channel , Histamine Receptor
T1257	Bestatin	Ubenimex	Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
	Bestatin (Ubenimex) competitively inhibits many aminopeptidases, including B, N and leucine aminopeptidases. Ubenimex is a microbial metabolite and dipeptide with potential immunomodulatory and antitumor activities. Amin...		Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
T1123	Camptothecin	NSC-100880,Campathecin,(S)-(+)-Camptothecin,CPT	Apoptosis , Influenza Virus , Topoisomerase , Antibiotic , Antifungal
	Camptothecin (CPT) belongs to the alkaloid group of natural products and is a specific DNA topoisomerase I (Topo I) inhibitor (IC50=679 nM) with specificity. Camptothecin has antitumor activity and induces apoptosis.
T25327	Didemnin B	NSC 325319,NSC325319,NSC-325319,Didemnin-B	Antiviral
	Didemnin B (Didemnin-B) is a depsipeptide extracted from the marine tunicate Trididemnin cyanophorum that has antiviral and antitumor activity.		Antiviral
T13476	β-Elemene	(-)-β-Elemene,Levo-β-elemene	Apoptosis
	β-Elemene (Levo-β-elemene) is a natural product isolated from Curcuma wenyujin, with an antitumor activity and induce cell apoptosis.		Apoptosis
T5237	Hexadecanedioic acid	1,14-Tetradecanedicarboxylic acid,1,16-Hexadecanedioic acid,Thapsic acid	Others , Endogenous Metabolite
	Hexadecanedioic acid (1,16-Hexadecanedioic acid) is a common saturated fatty acid found in animals, plants and microorganisms. It has antitumor activity.		Others , Endogenous Metabolite
T2920	Berbamine dihydrochloride	Berbamine,dihydrochloride	Apoptosis , NF-κB , Bcr-Abl , Autophagy
	Berbamine dihydrochloride (Berbamine), a natural compound derived from the Berberis amurensis plant, has been shown to exhibit antitumor activity in several Ys.		Apoptosis , NF-κB , Bcr-Abl , Autophagy
TN1010	Polyphyllin H		Others
	Polyphyllin H can be extracted from loblolly pine and rhizomes, has antitumor activity, and is used in studies of inflammation, fractures, and convulsions.		Others
TN7241	Annatto
	Annatto is a natural food coloring derived primarily from Bixa orellana L. Annatto has antitumor activity and at high doses increases the likelihood of cellular mutations.Annatto can be used in beverages, baking, and oth...
T13229	Tunicamycin		Influenza Virus , Antibacterial , Antibiotic , Antifungal
	Tunicamycin is a mixture of antibiotics that inhibit N-linked glycosylation by blocking GlcNAc phosphotransferase (GPT). Tunicamycin has antitumor activity, as well as anti-bacterial, anti-fungal, and anti-viral activity...		Influenza Virus , Antibacterial , Antibiotic , Antifungal
TN1049	Ingenol-5,20-acetonide		Others
	Ingenol-5,20-acetonide is a natural compound, an analog of Ingenol 3-Angelate. It has antitumor activity when used topically in the treatment of actinic keratoses.		Others
TN2326	(Z)-Butylidenephthalide	(Z)-3-Butylidenephthalide	Glucosidase
	(Z)-Butylidenephthalide ((Z)-3-Butylidenephthalide) has antitumor and hypoglycemic effects, and can effectively inhibit the tumor growth of glioma and inhibit R-glucosidase activity.		Glucosidase
T2908	Palmitic acid	Hexadecoic acid,hexadecanoic acid,Cetylic acid	HSP , Endogenous Metabolite
	Palmitic acid (Cetylic acid) is a natural product, a common saturated fatty acid found in animals, plants and microorganisms. Palmitic acid has antitumor activity.		HSP , Endogenous Metabolite
TQ0213	Bruceantin	(-)-Bruceantin,NCI165563,NSC165563	Others
			Others
T3519	Formosanin C	Polyphyllin B	Apoptosis , Caspase
	Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity in cultured cells and animal systems.		Apoptosis , Caspase
TN1369	Alloimperatorin	Prangenidin	Others
	Alloimperatorin (Prangenidin) exhibits in vitro antitumor activity in HL-60 acute myeloid leukemia cancer cells via inducing apoptosis, cell cycle disruption and inhibition of cell migration. It photosensitizes efficient...		Others
T4S0795	Berberrubine chloride	9-Berberoline Chloride,Beroline,Beroline Chloride,Berberrubine,9-Berberoline	IL Receptor
	1. Berberrubine chloride (9-Berberoline Chloride) has antitumor activity. 2. Berberrubine has antidiabetic activity. 3. Berberrubine dose-dependently inhibits IL-8 and MCP-1 protein levels in the media and mRNA expressio...		IL Receptor
TN3601	Carminic acid		ROS
	Carminic acid, the well-known red dyestuff from cochineal insects (Dactylopius spp.), is a potent feeding deterrent to ants. Carminic acid is an antioxidant to protect erythrocytes and DNA against radical-induced oxidati...		ROS
TN1047	Ingenol mebutate	Ingenol 3-Angelate,PEP005	gp120/CD4 , HIV Protease , PKC
	Ingenol mebutate (Ingenol 3-Angelate) is a potent activator of PKC subtypes including PKC-α, PKC-β, PKC-γ, PKC-δ, and PKC-ε with Kis of 0.3, 0.105, 0.162, 0.376, and 0.171 nM. Ingenol mebutate exhibits antiinflammatory a...		gp120/CD4 , HIV Protease , PKC
TQ0309	Glaucocalyxin B		Autophagy
			Autophagy
TN1258	3-Acetyl-beta-boswellic acid	3-O-Acetyl-beta-boswellic acid	DNA/RNA Synthesis
	3-Acetyl-beta-boswellic acid has antitumor activity, it inhibits synthesis of DNA, RNA and protein in human leukemia HL-60 cells in a dose dependent manner with IC50 values ranging from 0.6 to 7.1 microM.		DNA/RNA Synthesis
T6116	Bleomycin Sulfate	Blenoxane,NSC125066	DNA/RNA Synthesis , Antibiotic
	Bleomycin Sulfate (Blenoxane) is a glycopeptide antibiotic, an inhibitor of DNA synthesis. Bleomycin Sulfate causes DNA strand breaks but not RNA strand breaks. Bleomycin Sulfate has antitumor activity.		DNA/RNA Synthesis , Antibiotic
T4720	6-Hydroxypyridin-2(1H)-one hydrochloride	2,6-Dihydroxypyridine hydrochloride	Others , Endogenous Metabolite
	6-Hydroxypyridin-2(1H)-one hydrochloride (2,6-Dihydroxypyridine hydrochloride) is used as a reagent to synthesize uridine phosphorylase inhibitors that increase Uridine (Urd) (U829910) levels. Uridine is a promising bioc...		Others , Endogenous Metabolite
T8181	Poricoic acid A	Poricoic acid A(F)	Others
	Poricoic acid A (Poricoic acid A(F)) is a natural product with antitumor activity. It also enhances melatonin inhibition of AKI-to-CKD transition by regulating the Gas6/AxlNFκB/Nrf2 axis.		Others
TN1816	Kadsurin		Antioxidant
	Kadsurin has anti-oxidant activity, it induces enzymes capable of scavenging oxygen radical species in the liver. Kadsurin may be valuable antitumor promoters or chemopreventors.		Antioxidant
T3S1955	7-Ethylcamptothecin		Others
	1. 7-Ethylcamptothecin has the superior antitumor activity than CPT. (a). 7-Ethylcamptothecin has a stronger growth-inhibiting activity against tumor cells. (b). 7-Ethylcamptothecin remains in the intestinal tract for a ...		Others
T2219	Puromycin dihydrochloride	CL13900 dihydrochloride,Puromycin 2HCl	ribosome , DNA/RNA Synthesis , Antibacterial , Antibiotic
	Puromycin dihydrochloride (CL13900 dihydrochloride) is a cinnamamide adenosine antibiotic and an inhibitor of protein synthesis. Puromycin dihydrochloride inhibits protein synthesis by binding to RNA and has antitumor an...		ribosome , DNA/RNA Synthesis , Antibacterial , Antibiotic
T7452	2-methoxycinnamaldehyde	O-methoxycinnamaldehyde	Apoptosis , Others
	2-methoxycinnamaldehyde is a natural compound of Cinnamomum cassia,has been widely studied with regard to its antitumor activity.		Apoptosis , Others
T1272	Cytarabine	Ara-C,Cytosine Arabinoside,Cytosine β-D-arabinofuranoside,Arabinocytidine	Apoptosis , Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis , Endogenous Metabolite , Autophagy , HSV
	Cytarabine (Ara-C) is a nucleoside analog, an inhibitor of DNA synthesis (IC50=16 nM). Cytarabine inhibits DNA polymerase and induces cell cycle arrest, autophagy, and apoptosis. Cytarabine has antitumor activity.
T1521	(±)-10-Hydroxycamptothecin	Hydroxy Camptothecine,10-Hydroxycamptothecin	Topoisomerase
	(±)-10-Hydroxycamptothecin (Hydroxy Camptothecine) is an alkaloid isolated from the stem wood of the Chinese tree, Camptotheca acuminata. This compound selectively inhibits the nuclear enzyme DNA topoisomerase, type I. S...		Topoisomerase
T1703	SN-38	NK012,SN 38	DNA/RNA Synthesis , Topoisomerase , Autophagy
	SN-38 (NK012) is the active metabolite of Irinotecan, a DNA topoisomerase I (Topo I) inhibitor, which inhibits DNA and RNA synthesis (IC50=0.077/1.3 μM). SN-38 has antitumor activity and induces autophagy.		DNA/RNA Synthesis , Topoisomerase , Autophagy
T1181	Gefitinib	ZD1839	EGFR , Tyrosine Kinases , Autophagy
	Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 Del and L858R mutations. Gefitinib has antitumor activity and is used for the treatment of EGFR-mutated non-small-cell...		EGFR , Tyrosine Kinases , Autophagy
TWS1977	Kamebakaurin	Kamebakaurine	NF-κB
	1. Kamebakaurin (Kamebakaurine) has the ability to protect the liver from APAP-induced hepatotoxicity, presumably by both inhibiting the inflammatory response and oxidative stress. 2. Kamebakaurin inhibits the expression...		NF-κB
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天然物製品

Hypericin

T6S0923

Synonym: Hypericine,Cyclosan

Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC

2-Acetyl-3-ethylpyrazine

T67047

Synonym:

Target: Endogenous Metabolite

Palmaturbine

T3S1457

Synonym: Palmatrubin,Palmatrubine

Target: Others

4,6-Benzilidine-D-Glucose

Sodium Demethylcantharidate

T2736

Synonym: Sodium norcantharidin

Target: Others, Endogenous Metabolite

Torachrysone Triglucoside

TN7250

Synonym: 1-[8-[(O-β-D-Glucopyranosyl-(1→3)-O-β-D-glucopyranosyl-(1→6)-β-D-glucopyranosyl)oxy]-1-hydroxy-6-methoxy-3-methyl-2-naphthalenyl]ethanone

Target: Others

Doxycycline

T1687

Synonym: Vibramycin,Doxiciclina,Doxytetracycline,Doxycyclinum

Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite

6-(γ,γ-Dimethylallylamino)purine

T5581

Synonym: N6-(2-lsopentenyl)adenine,Triacanthine

Target: Others

Raddeanin A

T3878

Synonym: NSC382873,Anemodeanin A,Raddeanin R3

Target: Apoptosis, HDAC

Cephalomannine

T2217

Synonym: Baccatin III

Target: Microtubule Associated

Doxycycline (hyclate)

T1687L

Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,WC2031,Doxycycline hyclate

Target: MMP, ribosome, Antibacterial, Antibiotic

Synonym: Tenacissimoside C

Target: Others

Ursolic acid acetate

T3819

Synonym: Acetylursolic acid,3-Acetylursolic Acid

Target: AChE

Decitabine

T1508

Synonym: Dacogen,NSC 127716,Deoxycytidine,5-Aza-2'-deoxycytidine

Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA Methyltransferase

Testosterone acetate

TC0025

Synonym: NSC523836,NSC-523836,NSC 523836

Target: CaMK, Calcium Channel, Histamine Receptor

Bestatin

T1257

Synonym: Ubenimex

Target: Others, Aminopeptidase, Antibacterial, Antibiotic, LTR

Camptothecin

T1123

Synonym: NSC-100880,Campathecin,(S)-(+)-Camptothecin,CPT

Target: Apoptosis, Influenza Virus, Topoisomerase, Antibiotic, Antifungal

Didemnin B

T25327

Synonym: NSC 325319,NSC325319,NSC-325319,Didemnin-B

Target: Antiviral

β-Elemene

T13476

Synonym: (-)-β-Elemene,Levo-β-elemene

Target: Apoptosis

Hexadecanedioic acid

T5237

Synonym: 1,14-Tetradecanedicarboxylic acid,1,16-Hexadecanedioic acid,Thapsic acid

Target: Others, Endogenous Metabolite

Berbamine dihydrochloride

T2920

Synonym: Berbamine,dihydrochloride

Target: Apoptosis, NF-κB, Bcr-Abl, Autophagy

Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal

Ingenol-5,20-acetonide

TN1049

Synonym:

Target: Others

(Z)-Butylidenephthalide

TN2326

Synonym: (Z)-3-Butylidenephthalide

Target: Glucosidase

Palmitic acid

T2908

Synonym: Hexadecoic acid,hexadecanoic acid,Cetylic acid

Target: HSP, Endogenous Metabolite

Bruceantin

TQ0213

Synonym: (-)-Bruceantin,NCI165563,NSC165563

Target: Others

Formosanin C

T3519

Synonym: Polyphyllin B

Target: Apoptosis, Caspase

Berberrubine chloride

T4S0795

Synonym: 9-Berberoline Chloride,Beroline,Beroline Chloride,Berberrubine,9-Berberoline

Synonym: Ingenol 3-Angelate,PEP005

Target: gp120/CD4, HIV Protease, PKC

3-Acetyl-beta-boswellic acid

TN1258

Synonym: 3-O-Acetyl-beta-boswellic acid

Target: DNA/RNA Synthesis

Bleomycin Sulfate

T6116

Synonym: Blenoxane,NSC125066

Target: DNA/RNA Synthesis, Antibiotic

6-Hydroxypyridin-2(1H)-one hydrochloride

T4720

Synonym: 2,6-Dihydroxypyridine hydrochloride

Target: Others, Endogenous Metabolite

Poricoic acid A

T8181

Synonym: Poricoic acid A(F)

Puromycin dihydrochloride

T2219

Synonym: CL13900 dihydrochloride,Puromycin 2HCl

Target: ribosome, DNA/RNA Synthesis, Antibacterial, Antibiotic

2-methoxycinnamaldehyde

T7452

Synonym: O-methoxycinnamaldehyde

Target: Apoptosis, Others

Cytarabine

T1272

Synonym: Ara-C,Cytosine Arabinoside,Cytosine β-D-arabinofuranoside,Arabinocytidine

Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy, HSV

(±)-10-Hydroxycamptothecin

T1521

Synonym: Hydroxy Camptothecine,10-Hydroxycamptothecin

Target: Topoisomerase

SN-38

T1703

Synonym: NK012,SN 38

Target: DNA/RNA Synthesis, Topoisomerase, Autophagy

Gefitinib

T1181

Synonym: ZD1839

Target: EGFR, Tyrosine Kinases, Autophagy

Kamebakaurin

TWS1977

Synonym: Kamebakaurine

Target: NF-κB

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-06983	IFN gamma Protein, Human, Recombinant (E. coli)	Human	E. coli
	IFN gamma, also known as IFNG, is a secreted protein that belongs to the type II interferon family. IFN gamma is produced predominantly by natural killer and natural killer T cells as part of the innate immune response, ...
TMPH-03055	Ribonuclease mitogillin Protein, Neosartorya fumigata, Recombinant (His & Myc & SUMO)	Neosartorya fumigata	E. coli
	This purine-specific ribonuclease cleaves 28S RNA in eukaryotic ribosomes, inhibits protein synthesis, and shows antitumor activity.
TMPH-00131	Ribonuclease mitogillin Protein, Aspergillus restrictus, Recombinant (His & Myc)	Aspergillus restrictus	E. coli
	This purine-specific ribonuclease cleaves 28S RNA in eukaryotic ribosomes, inhibits protein synthesis, and shows antitumor activity. Ribonuclease mitogillin Protein, Aspergillus restrictus, Recombinant (His & Myc) is exp...
TMPJ-00008	CXCL10 Protein, Human, Recombinant (hFc & His)	Human	HEK293 Cells
	Human C-X-C Motif Chemokine Ligand 10 (CXCL10) is a non-ELR chemokine secreted by various cell types, such as monocytes, endothelial cells and fibroblasts, in response to IFN-γ. CXCL10 functions via chemokine receptor CX...
TMPH-02451	IFN gamma Protein, Marmota monax, Recombinant (His)	Marmota monax	P. pastoris (Yeast)
	Produced by lymphocytes activated by specific antigens or mitogens. IFN-gamma, in addition to having antiviral activity, has important immunoregulatory functions. It is a potent activator of macrophages, it has antiproli...
TMPJ-00076	IL-28B Protein, Human, Recombinant	Human	HEK293 Cells
	Interleukin-28B, also known as Cytokine Zcyto22, Interferon lambda-3, Interferon lambda-4, IFNL3, IFNL4, ZCYTO22 and IL28B, is a secreted cytokine which belongs to the IL-28/IL-29 family. IL-28 has also been shown to pla...
TMPH-00373	IFN gamma Protein, Chicken, Recombinant (GST)	Chicken	E. coli
	Produced by lymphocytes activated by specific antigens or mitogens. IFN-gamma, in addition to having antiviral activity, has important immunoregulatory functions. It is a potent activator of macrophages, it has antiproli...

IFN gamma Protein, Human, Recombinant (E. coli)

TMPY-06983

Species: Human

Expression System: E. coli

Ribonuclease mitogillin Protein, Neosartorya fumigata, Recombinant (His & Myc & SUMO)

TMPH-03055

Species: Neosartorya fumigata

Expression System: E. coli

Ribonuclease mitogillin Protein, Aspergillus restrictus, Recombinant (His & Myc)

TMPH-00131

Species: Aspergillus restrictus

Expression System: E. coli

CXCL10 Protein, Human, Recombinant (hFc & His)

TMPJ-00008

Species: Human

Expression System: HEK293 Cells

IFN gamma Protein, Marmota monax, Recombinant (His)

TMPH-02451

Species: Marmota monax

Expression System: P. pastoris (Yeast)

IL-28B Protein, Human, Recombinant

TMPJ-00076

Species: Human

Expression System: HEK293 Cells

IFN gamma Protein, Chicken, Recombinant (GST)

TMPH-00373

Species: Chicken

Expression System: E. coli

カタログ番号	製品名
L6700	Anti-Tumor Natural Product Library	1772 compounds
	A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L9300	Macrocyclic Compound Library	210 compounds
	210 macrocyclic compounds of known activity for high-throughput, high-content screening;

ライブラリー

Anti-Tumor Natural Product Library

L6700

Compounds: 1772

Macrocyclic Compound Library

L9300

Compounds: 210